Didesmethyl cariprazine is a metabolite of Cariprazine and acts as the predominant circulating active moiety. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a antipsychotic agent candidate that exhibits high affinity for the D 3 and D 2 receptors, and moderate affinity for the 5-HT 1A receptor
IC50& Target:5-HT 1A Receptor D 3 Receptor D 2 Receptor
规格
别名
二去甲基卡利拉嗪
规格或纯度
10mM in DMSO
英文名称
Didesmethyl cariprazine
生化机理
双甲基卡哌嗪是卡哌嗪的代谢物,是主要的循环活性分子。双甲基卡哌嗪的半衰期较长,为 1-3 周。卡利普嗪是一种抗精神病候选药物,对 D 3