α-Glucosidase-IN-68 (Compound 2) is an inhibitor for α-Glucosidase , AChE , and BChE , with IC 50 of 0.251, 0.774 and 0.793 μM, respectively. α-Glucosidase-IN-68 exhibits antioxidant efficacy, with IC 50 of 0.69 μM and 0.02 μM, in DPPH and ABTS experiments. α-Glucosidase-IN-68 exhibits antidiabetic effect in Streptozotocin -induced diabetic rat models.