(R)-MLN-4760, the R-enantiomer of MLN-4760, is an ACE2 inhibitor, with an IC 50 of 8.4 μM. (R)-MLN-4760 is the less active isomer
In Vitro
(R)-MLN-4760 (compound 16RS) is the less active isomer of MLN-4760. MCE has not independently confirmed the accuracy of these methods. They are for reference only.