MAC glucuronide alpha hydroxy lactone linked SN-38 is a stable lactone compound composed of ADC toxin SN-38 (Topoisomerase I inhibitor) and MAC glucuronide alpha hydroxy lactone. MAC glucuronide α - hydroxy lactone linked SN-38 exhibits cytotoxicity towards L540cy cells and Ramos cells, with IC50 values of 99 and 105 ng/mL, respectively.
规格
英文名称
MAC glucuronide α-hydroxy lactone-linked SN-38
生化机理
MAC glucuronide α-hydroxy lactone-linked SN-38 (Topoisomerase I inhibitor) is a stabilized lactone MAC glucuronide α-hydroxy lactone-linked SN-38 agent linker. MAC glucuronide α-hydroxy lactone-linked SN-38 is cytotoxic across L540cy cells and Ramos cells with IC50 values of 99 and 105 ng/mL, respectively.