ATR-IN-4 is a potent ATR (Ataxia telangiectasia mutated gene Rad 3-associated kinase) inhibitor. ATR-IN-4 inhibits growth of human prostate cancer cells DU145 and human lung cancer cells NCI-H460 with IC 50 s of 130.9 nM and 41.33 nM, respectively. (Patent CN112142744A, compound 13).
Form:Solid
规格
规格或纯度
≥99%
英文名称
ATR-IN-4
生化机理
ATR-IN-4 是一种强效的 ATR(共济失调毛细血管扩张症突变基因 Rad 3 相关激酶)抑制剂。ATR-IN-4 可抑制人前列腺癌细胞 DU145 和人肺癌细胞 NCI-H460 的生长,其 IC 50 s 分别为 130.9 nM 和 41 .33 nM。(贝特