浏览与蛋白激酶靶点相关的小分子及工具化合物,用于激酶生物学、筛选及通路研究。本页面可帮助您比较药物发现研究中最受关注的靶点类别之一中的抑制剂及相关调节剂。
蛋白激酶(Protein kinases)
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丝裂原活化蛋白激酶1(MAPK1) Mitogen-activated protein kinase 1 (MAPK1)
1,681丙酮酸激酶 pkm (PKM) Pyruvate kinase pkm (PKM)
594丝氨酸蛋白激酶 atm (ATM) Serine-protein kinase atm (ATM)
315表皮生长因子受体(EGFR) Epidermal growth factor receptor (EGFR)
535糖原合成酶激酶-3β (GSK3B) Glycogen synthase kinase-3 beta (GSK3B)
325细胞周期蛋白依赖性激酶2 (CDK2) Cyclin-dependent kinase 2 (CDK2)
321血管内皮生长因子受体 2 (KDR) Vascular endothelial growth factor receptor 2 (KDR)
363酪氨酸蛋白激酶 lck (LCK) Tyrosine-protein kinase lck (LCK)
244原癌基因酪氨酸蛋白激酶 src (SRC) Proto-oncogene tyrosine-protein kinase src (SRC)
292受体型酪氨酸蛋白激酶 flt3 (FLT3) Receptor-type tyrosine-protein kinase flt3 (FLT3)
303丝裂原活化蛋白激酶14 (MAPK14) Mitogen-activated protein kinase 14 (MAPK14)
196成纤维细胞生长因子受体 1 (FGFR1) Fibroblast growth factor receptor 1 (FGFR1)
137丝裂原活化蛋白激酶 10 (MAPK10) Mitogen-activated protein kinase 10 (MAPK10)
94极光激酶A(AURKA) Aurora kinase a (AURKA)
173酪氨酸蛋白激酶 abl1 (ABL1) Tyrosine-protein kinase abl1 (ABL1)
190细胞周期蛋白依赖性激酶5 (CDK5) Cyclin-dependent-like kinase 5 (CDK5)
119丝氨酸/苏氨酸蛋白激酶 pim-1 (PIM1) Serine/threonine-protein kinase pim-1 (PIM1)
101双特异性酪氨酸磷酸化调节激酶 1a (DYRK1A) Dual specificity tyrosine-phosphorylation-regulated kinase 1a (DYRK1A)
157细胞周期蛋白依赖性激酶1(CDK1) Cyclin-dependent kinase 1 (CDK1)
152Rac-α丝氨酸/苏氨酸蛋白激酶(AKT1) Rac-alpha serine/threonine-protein kinase (AKT1)
99丝氨酸/苏氨酸蛋白激酶 mTOR (MTOR) Serine/threonine-protein kinase mtor (MTOR)
425酪氨酸蛋白激酶 JAK2 (JAK2) Tyrosine-protein kinase jak2 (JAK2)
219极光激酶b(AURKB) Aurora kinase b (AURKB)
137丝氨酸/苏氨酸蛋白激酶 chk1 (CHEK1) Serine/threonine-protein kinase chk1 (CHEK1)
73肝细胞生长因子受体(MET) Hepatocyte growth factor receptor (MET)
142糖原合成酶激酶-3α (GSK3A) Glycogen synthase kinase-3 alpha (GSK3A)
74酪氨酸蛋白激酶 fyn (FYN) Tyrosine-protein kinase fyn (FYN)
189胰岛素样生长因子1受体(IGF1R) Insulin-like growth factor 1 receptor (IGF1R)
70酪氨酸蛋白激酶 btk (BTK) Tyrosine-protein kinase btk (BTK)
154丝裂原活化蛋白激酶 8 (MAPK8) Mitogen-activated protein kinase 8 (MAPK8)
59原癌基因酪氨酸蛋白激酶受体 RET (RET) Proto-oncogene tyrosine-protein kinase receptor ret (RET)
118Rho相关蛋白激酶1(ROCK1) Rho-associated protein kinase 1 (ROCK1)
87胰岛素受体(INSR) Insulin receptor (INSR)
40蛋白酪氨酸激酶2β(PTK2B) Protein-tyrosine kinase 2-beta (PTK2B)
44Rho相关蛋白激酶2(ROCK2) Rho-associated protein kinase 2 (ROCK2)
101高亲和力神经生长因子受体(NTRK1) High affinity nerve growth factor receptor (NTRK1)
107丝裂原活化蛋白激酶9 (MAPK9) Mitogen-activated protein kinase 9 (MAPK9)
47非受体酪氨酸蛋白激酶 tyk2 (TYK2) Non-receptor tyrosine-protein kinase tyk2 (TYK2)
127细胞周期蛋白依赖性激酶9 (CDK9) Cyclin-dependent kinase 9 (CDK9)
141血小板衍生生长因子受体β(PDGFRB) Platelet-derived growth factor receptor beta (PDGFRB)
151核糖体蛋白S6激酶α-3(RPS6KA3) Ribosomal protein s6 kinase alpha-3 (RPS6KA3)
38黏着斑激酶1(PTK2) Focal adhesion kinase 1 (PTK2)
69rac-β丝氨酸/苏氨酸蛋白激酶(AKT2) Rac-beta serine/threonine-protein kinase (AKT2)
51依赖营地的蛋白激酶催化亚基α(PRKACA) Camp-dependent protein kinase catalytic subunit alpha (PRKACA)
32Lim结构域激酶1(LIMK1) Lim domain kinase 1 (LIMK1)
50酪蛋白激酶 I 亚型 α (CSNK1A1) Casein kinase i isoform alpha (CSNK1A1)
38MAP激酶激活蛋白激酶2 (MAPKAPK2) Map kinase-activated protein kinase 2 (MAPKAPK2)
46丝氨酸/苏氨酸蛋白激酶 PAK4 (PAK4) Serine/threonine-protein kinase pak 4 (PAK4)
22酪蛋白激酶 I 同工型 δ (CSNK1D) Casein kinase i isoform delta (CSNK1D)
59酪氨酸蛋白激酶 syk (SYK) Tyrosine-protein kinase syk (SYK)
53蛋白激酶cδ型(PRKCD) Protein kinase c delta type (PRKCD)
435'-AMP激活蛋白激酶催化亚基α-1(PRKAA1) 5'-AMP-activated protein kinase catalytic subunit alpha-1 (PRKAA1)
28γ-丝氨酸/苏氨酸蛋白激酶(AKT3) Rac-gamma serine/threonine-protein kinase (AKT3)
40丝裂原活化蛋白激酶激酶激酶激酶4 (MAP4K4) Mitogen-activated protein kinase kinase kinase kinase 4 (MAP4K4)
33丝氨酸/苏氨酸蛋白激酶 nek2 (NEK2) Serine/threonine-protein kinase nek2 (NEK2)
14丝氨酸/苏氨酸蛋白激酶 plk1 (PLK1) Serine/threonine-protein kinase plk1 (PLK1)
82酪氨酸蛋白激酶 JAK3 (JAK3) Tyrosine-protein kinase jak3 (JAK3)
173酪氨酸蛋白激酶 lyn (LYN) Tyrosine-protein kinase lyn (LYN)
31双特异性蛋白激酶 clk2 (CLK2) Dual specificity protein kinase clk2 (CLK2)
57白细胞介素-1受体相关激酶4(IRAK4) Interleukin-1 receptor-associated kinase 4 (IRAK4)
47双特异性丝裂原活化蛋白激酶激酶1 (MAP2K1) Dual specificity mitogen-activated protein kinase kinase 1 (MAP2K1)
86双特异性蛋白激酶 clk4 (CLK4) Dual specificity protein kinase clk4 (CLK4)
92细胞周期蛋白依赖性激酶 4 (CDK4) Cyclin-dependent kinase 4 (CDK4)
104丝裂原活化蛋白激酶激酶激酶激酶2 (MAP4K2) Mitogen-activated protein kinase kinase kinase kinase 2 (MAP4K2)
17细胞周期蛋白依赖性激酶7 (CDK7) Cyclin-dependent kinase 7 (CDK7)
68核糖体蛋白S6激酶β-1(RPS6KB1) Ribosomal protein s6 kinase beta-1 (RPS6KB1)
36丝氨酸/苏氨酸蛋白激酶d3(PRKD3) Serine/threonine-protein kinase d3 (PRKD3)
17酪氨酸蛋白激酶 JAK1 (JAK1) Tyrosine-protein kinase jak1 (JAK1)
138Ephrin a 型受体 2 (EPHA2) Ephrin type-a receptor 2 (EPHA2)
18丝氨酸/苏氨酸蛋白激酶 tao1 (TAOK1) Serine/threonine-protein kinase tao1 (TAOK1)
23Map/微管亲和力调节激酶3 (MARK3) Map/microtubule affinity-regulating kinase 3 (MARK3)
22丝氨酸/苏氨酸蛋白激酶3 (STK3) Serine/threonine-protein kinase 3 (STK3)
11丝氨酸/苏氨酸蛋白激酶 plk4 (PLK4) Serine/threonine-protein kinase plk4 (PLK4)
33丝氨酸/苏氨酸蛋白激酶d2 (PRKD2) Serine/threonine-protein kinase d2 (PRKD2)
22丝氨酸/苏氨酸蛋白激酶 BRAF (BRAF) Serine/threonine-protein kinase b-raf (BRAF)
96丝氨酸/苏氨酸蛋白激酶n2 (PKN2) Serine/threonine-protein kinase n2 (PKN2)
17磷脂酰肌醇 4,5-二磷酸 3-激酶催化亚基 α 同工型 (PIK3CA) Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PIK3CA)
323丝氨酸/苏氨酸蛋白激酶 mrck alpha (CDC42BPA) Serine/threonine-protein kinase mrck alpha (CDC42BPA)
9双特异性蛋白激酶 clk1 (CLK1) Dual specificity protein kinase clk1 (CLK1)
103白细胞介素-1受体相关激酶1(IRAK1) Interleukin-1 receptor-associated kinase 1 (IRAK1)
22肥大细胞/干细胞生长因子受体试剂盒(KIT) Mast/stem cell growth factor receptor kit (KIT)
175母体胚胎亮氨酸拉链激酶(MELK) Maternal embryonic leucine zipper kinase (MELK)
28受体酪氨酸蛋白激酶 erbb-2 (ERBB2) Receptor tyrosine-protein kinase erbb-2 (ERBB2)
128钙/钙调蛋白依赖性蛋白激酶II型亚基δ(CAMK2D) Calcium/calmodulin-dependent protein kinase type ii subunit delta (CAMK2D)
17丝裂原活化蛋白激酶激酶激酶 mlt (ZAK) Mitogen-activated protein kinase kinase kinase mlt (ZAK)
12蛋白激酶cα型(PRKCA) Protein kinase c alpha type (PRKCA)
71丝氨酸/苏氨酸蛋白激酶mark2(MARK2) Serine/threonine-protein kinase mark2 (MARK2)
31丝裂原活化蛋白激酶激酶激酶激酶 5 (MAP4K5) Mitogen-activated protein kinase kinase kinase kinase 5 (MAP4K5)
22核糖体蛋白S6激酶α-5(RPS6KA5) Ribosomal protein s6 kinase alpha-5 (RPS6KA5)
16核因子κB激酶亚基ε抑制剂(IKBKE) Inhibitor of nuclear factor kappa-b kinase subunit epsilon (IKBKE)
23Ste20样丝氨酸/苏氨酸蛋白激酶(SLK) Ste20-like serine/threonine-protein kinase (SLK)
7活化的 cdc42 激酶 1 (TNK2) Activated cdc42 kinase 1 (TNK2)
28磷酸化酶b激酶γ催化链,肝/睾丸同工型(PHKG2) Phosphorylase b kinase gamma catalytic chain, liver/testis isoform (PHKG2)
0蛋白激酶cθ型(PRKCQ) Protein kinase c theta type (PRKCQ)
44蛋白酪氨酸激酶 6 (PTK6) Protein-tyrosine kinase 6 (PTK6)
16丝氨酸/苏氨酸蛋白激酶 pim-2 (PIM2) Serine/threonine-protein kinase pim-2 (PIM2)
39激活素受体1型(ACVR1) Activin receptor type-1 (ACVR1)
46钙/钙调蛋白依赖性蛋白激酶II型亚基γ(CAMK2G) Calcium/calmodulin-dependent protein kinase type ii subunit gamma (CAMK2G)
2MAP激酶激活蛋白激酶5 (MAPKAPK5) Map kinase-activated protein kinase 5 (MAPKAPK5)
15巨噬细胞集落刺激因子1受体(CSF1R) Macrophage colony-stimulating factor 1 receptor (CSF1R)
134丝氨酸/苏氨酸蛋白激酶 tbk1 (TBK1) Serine/threonine-protein kinase tbk1 (TBK1)
39酪蛋白激酶 I 同工型 γ-1 (CSNK1G1) Casein kinase i isoform gamma-1 (CSNK1G1)
5Cgmp依赖性蛋白激酶1(PRKG1) Cgmp-dependent protein kinase 1 (PRKG1)
12TGF-β受体1型(TGFBR1) Tgf-beta receptor type-1 (TGFBR1)
91巨噬细胞刺激蛋白受体(MST1R) Macrophage-stimulating protein receptor (MST1R)
18蛋白激酶c Iota型(PRKCI) Protein kinase c iota type (PRKCI)
17酪蛋白激酶 I 同工型 γ-3 (CSNK1G3) Casein kinase i isoform gamma-3 (CSNK1G3)
2酪氨酸蛋白激酶 fer (FER) Tyrosine-protein kinase fer (FER)
16ALK酪氨酸激酶受体(ALK) Alk tyrosine kinase receptor (ALK)
84酪氨酸蛋白激酶 frk (FRK) Tyrosine-protein kinase frk (FRK)
6丝裂原活化蛋白激酶3 (MAPK3) Mitogen-activated protein kinase 3 (MAPK3)
50酪氨酸蛋白激酶 fes/fps (FES) Tyrosine-protein kinase fes/fps (FES)
8双特异性丝裂原活化蛋白激酶激酶2 (MAP2K2) Dual specificity mitogen-activated protein kinase kinase 2 (MAP2K2)
40酪蛋白激酶 I 同工酶 ε (CSNK1E) Casein kinase i isoform epsilon (CSNK1E)
41磷脂酰肌醇 4,5-二磷酸 3-激酶催化亚基γ同工型 (PIK3CG) Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (PIK3CG)
248酪蛋白激酶 I 同工型 γ-2 (CSNK1G2) Casein kinase i isoform gamma-2 (CSNK1G2)
4丝氨酸/苏氨酸蛋白激酶/核糖核酸内切酶ire1 (ERN1) Serine/threonine-protein kinase/endoribonuclease ire1 (ERN1)
63血管内皮生长因子受体 1 (FLT1) Vascular endothelial growth factor receptor 1 (FLT1)
89丝裂原活化蛋白激酶激酶激酶 5 (MAP3K5) Mitogen-activated protein kinase kinase kinase 5 (MAP3K5)
28Ephrin B 型受体 4 (EPHB4) Ephrin type-b receptor 4 (EPHB4)
12酪氨酸蛋白激酶是(YES1) Tyrosine-protein kinase yes (YES1)
47核糖体蛋白S6激酶α-1(RPS6KA1) Ribosomal protein s6 kinase alpha-1 (RPS6KA1)
34Wee1样蛋白激酶(WEE1) Wee1-like protein kinase (WEE1)
20受体相互作用丝氨酸/苏氨酸蛋白激酶 2 (RIPK2) Receptor-interacting serine/threonine-protein kinase 2 (RIPK2)
67上皮盘状结构域受体 1 (DDR1) Epithelial discoidin domain-containing receptor 1 (DDR1)
72丝裂原活化蛋白激酶11 (MAPK11) Mitogen-activated protein kinase 11 (MAPK11)
45酪氨酸蛋白激酶 hck (HCK) Tyrosine-protein kinase hck (HCK)
18蛋白激酶cβ型(PRKCB) Protein kinase c beta type (PRKCB)
47酪氨酸蛋白激酶 csk (CSK) Tyrosine-protein kinase csk (CSK)
7Ephrin B 型受体 2 (EPHB2) Ephrin type-b receptor 2 (EPHB2)
11酪氨酸蛋白激酶 tec (TEC) Tyrosine-protein kinase tec (TEC)
47细胞周期蛋白依赖性激酶 6 (CDK6) Cyclin-dependent kinase 6 (CDK6)
46盘状结构域受体 2 (DDR2) Discoidin domain-containing receptor 2 (DDR2)
32细胞周期 g 相关激酶 (GAK) Cyclin-g-associated kinase (GAK)
55平滑肌肌球蛋白轻链激酶 (MYLK) Myosin light chain kinase, smooth muscle (MYLK)
22磷脂酰肌醇 4,5-二磷酸 3-激酶催化亚基δ同工型 (PIK3CD) Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform (PIK3CD)
241Lim结构域激酶2(LIMK2) Lim domain kinase 2 (LIMK2)
24丝氨酸/苏氨酸蛋白激酶n1(PKN1) Serine/threonine-protein kinase n1 (PKN1)
11钙/钙调蛋白依赖性蛋白激酶激酶2 (CAMKK2) Calcium/calmodulin-dependent protein kinase kinase 2 (CAMKK2)
8β-肾上腺素能受体激酶1(ADRBK1) Beta-adrenergic receptor kinase 1 (ADRBK1)
28丝裂原活化蛋白激酶激酶激酶11 (MAP3K11) Mitogen-activated protein kinase kinase kinase 11 (MAP3K11)
12丝氨酸/苏氨酸蛋白激酶 4 (STK4) Serine/threonine-protein kinase 4 (STK4)
12酪蛋白激酶 II 亚基 α' (CSNK2A2) Casein kinase II subunit alpha' (CSNK2A2)
23丝氨酸/苏氨酸蛋白激酶 sik2 (SIK2) Serine/threonine-protein kinase sik2 (SIK2)
153-磷酸肌醇依赖性蛋白激酶1(PDPK1) 3-phosphoinositide-dependent protein kinase 1 (PDPK1)
61激活素受体1b型(ACVR1B) Activin receptor type-1b (ACVR1B)
19Bdnf/nt-3 生长因子受体 (NTRK2) Bdnf/nt-3 growth factors receptor (NTRK2)
54骨形态发生蛋白受体1a型(BMPR1A) Bone morphogenetic protein receptor type-1a (BMPR1A)
24酪蛋白激酶 II 亚基 α (CSNK2A1) Casein kinase II subunit alpha (CSNK2A1)
75磷脂酰肌醇 4,5-二磷酸 3-激酶催化亚基 β 同工型 (PIK3CB) Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform (PIK3CB)
197Ap2 相关蛋白激酶 1 (AAK1) Ap2-associated protein kinase 1 (AAK1)
74Ephrin a 型受体 4 (EPHA4) Ephrin type-a receptor 4 (EPHA4)
4核糖体蛋白S6激酶α-4(RPS6KA4) Ribosomal protein s6 kinase alpha-4 (RPS6KA4)
4血管内皮生长因子受体3(FLT4) Vascular endothelial growth factor receptor 3 (FLT4)
66Abelson酪氨酸蛋白激酶2 (ABL2) Abelson tyrosine-protein kinase 2 (ABL2)
26丝氨酸/苏氨酸蛋白激酶 26 (MST4) Serine/threonine-protein kinase 26 (MST4)
7蛋白激酶c zeta型(PRKCZ) Protein kinase c zeta type (PRKCZ)
10BMP-2诱导蛋白激酶(BMP2K) Bmp-2-inducible protein kinase (BMP2K)
16骨形态发生蛋白受体1b型(BMPR1B) Bone morphogenetic protein receptor type-1b (BMPR1B)
17骨形态发生蛋白受体2型(BMPR2) Bone morphogenetic protein receptor type-2 (BMPR2)
5核糖体蛋白S6激酶α-6(RPS6KA6) Ribosomal protein s6 kinase alpha-6 (RPS6KA6)
7丝氨酸/苏氨酸蛋白激酶10 (STK10) Serine/threonine-protein kinase 10 (STK10)
11丝氨酸/苏氨酸蛋白激酶16 (STK16) Serine/threonine-protein kinase 16 (STK16)
10膜相关酪氨酸和苏氨酸特异性 cdc2 抑制激酶 (PKMYT1) Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase (PKMYT1)
9丝氨酸/苏氨酸蛋白激酶 nek1 (NEK1) Serine/threonine-protein kinase nek1 (NEK1)
4双特异性丝裂原活化蛋白激酶激酶 6 (MAP2K6) Dual specificity mitogen-activated protein kinase kinase 6 (MAP2K6)
2Ephrin B 型受体 3 (EPHB3) Ephrin type-b receptor 3 (EPHB3)
2血小板衍生生长因子受体α(PDGFRA) Platelet-derived growth factor receptor alpha (PDGFRA)
107TGF-β受体2型(TGFBR2) Tgf-beta receptor type-2 (TGFBR2)
22钙/钙调蛋白依赖性蛋白激酶IV型(CAMK4) Calcium/calmodulin-dependent protein kinase type iv (CAMK4)
2细胞分裂周期7相关蛋白激酶(CDC7) Cell division cycle 7-related protein kinase (CDC7)
26细胞周期蛋白依赖性激酶16 (CDK16) Cyclin-dependent kinase 16 (CDK16)
15细胞周期蛋白依赖性激酶13 (CDK13) Cyclin-dependent kinase 13 (CDK13)
22双特异性丝裂原活化蛋白激酶激酶3 (MAP2K3) Dual specificity mitogen-activated protein kinase kinase 3 (MAP2K3)
2丝氨酸/苏氨酸蛋白激酶 tao3 (TAOK3) Serine/threonine-protein kinase tao3 (TAOK3)
25Traf2 和 nck 相互作用蛋白激酶 (TNIK) Traf2 and nck-interacting protein kinase (TNIK)
12激活素受体2b型(ACVR2B) Activin receptor type-2b (ACVR2B)
10Ephrin a 型受体 5 (EPHA5) Ephrin type-a receptor 5 (EPHA5)
1畸形样激酶 1 (MINK1) Misshapen-like kinase 1 (MINK1)
21丝裂原活化蛋白激酶15 (MAPK15) Mitogen-activated protein kinase 15 (MAPK15)
6丝裂原活化蛋白激酶激酶激酶激酶3 (MAP4K3) Mitogen-activated protein kinase kinase kinase kinase 3 (MAP4K3)
7非受体酪氨酸蛋白激酶 tnk1 (TNK1) Non-receptor tyrosine-protein kinase tnk1 (TNK1)
16丝氨酸/苏氨酸蛋白激酶 ULK1 (ULK1) Serine/threonine-protein kinase ulk1 (ULK1)
17依赖营地的蛋白激酶催化亚基β(PRKACB) Camp-dependent protein kinase catalytic subunit beta (PRKACB)
6双特异性酪氨酸磷酸化调节激酶1b (DYRK1B) Dual specificity tyrosine-phosphorylation-regulated kinase 1b (DYRK1B)
73丝裂原活化蛋白激酶7 (MAPK7) Mitogen-activated protein kinase 7 (MAPK7)
21丝裂原活化蛋白激酶激酶激酶激酶1 (MAP4K1) Mitogen-activated protein kinase kinase kinase kinase 1 (MAP4K1)
12丝氨酸/苏氨酸蛋白激酶 tao2 (TAOK2) Serine/threonine-protein kinase tao2 (TAOK2)
26非典型激酶 adck3,线粒体 (ADCK3) Atypical kinase adck3, mitochondrial (ADCK3)
2柠檬酸rho相互作用激酶(CIT) Citron rho-interacting kinase (CIT)
6细胞周期蛋白依赖性激酶 12 (CDK12) Cyclin-dependent kinase 12 (CDK12)
38细胞周期蛋白依赖性激酶3 (CDK3) Cyclin-dependent kinase 3 (CDK3)
10丝裂原活化蛋白激酶激酶激酶1 (MAP3K1) Mitogen-activated protein kinase kinase kinase 1 (MAP3K1)
4丝裂原活化蛋白激酶激酶激酶2 (MAP3K2) Mitogen-activated protein kinase kinase kinase 2 (MAP3K2)
4磷脂酰肌醇 5-磷酸 4-激酶 2 型 γ (PIP4K2C) Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma (PIP4K2C)
12丝氨酸/苏氨酸蛋白激酶 nek9 (NEK9) Serine/threonine-protein kinase nek9 (NEK9)
4丝氨酸/苏氨酸蛋白激酶 nlk (NLK) Serine/threonine-protein kinase nlk (NLK)
7丝氨酸/苏氨酸蛋白激酶 sik3 (SIK3) Serine/threonine-protein kinase sik3 (SIK3)
12双特异性丝裂原活化蛋白激酶激酶 5 (MAP2K5) Dual specificity mitogen-activated protein kinase kinase 5 (MAP2K5)
19丝氨酸/苏氨酸蛋白激酶 lats1 (LATS1) Serine/threonine-protein kinase lats1 (LATS1)
1丝氨酸/苏氨酸蛋白激酶 mrck beta (CDC42BPB) Serine/threonine-protein kinase mrck beta (CDC42BPB)
0丝氨酸/苏氨酸蛋白激酶 ULK3 (ULK3) Serine/threonine-protein kinase ulk3 (ULK3)
0白细胞介素-1受体相关激酶3(IRAK3) Interleukin-1 receptor-associated kinase 3 (IRAK3)
4Nuak家族snf1样激酶2(NUAK2) Nuak family snf1-like kinase 2 (NUAK2)
16丝裂原活化蛋白激酶激酶激酶4 (MAP3K4) Mitogen-activated protein kinase kinase kinase 4 (MAP3K4)
0真核翻译起始因子2-α激酶1(EIF2AK1) Eukaryotic translation initiation factor 2-alpha kinase 1 (EIF2AK1)
11丝裂原活化蛋白激酶激酶激酶3 (MAP3K3) Mitogen-activated protein kinase kinase kinase 3 (MAP3K3)
0丝氨酸/苏氨酸蛋白激酶 nek3 (NEK3) Serine/threonine-protein kinase nek3 (NEK3)
1核因子κB激酶β亚基抑制剂(IKBKB) Inhibitor of nuclear factor kappa-b kinase subunit beta (IKBKB)
75Map/微管亲和力调节激酶4 (MARK4) Map/microtubule affinity-regulating kinase 4 (MARK4)
12Ephrin B 型受体 6 (EPHB6) Ephrin type-b receptor 6 (EPHB6)
10丝氨酸/苏氨酸蛋白激酶 PAK 2 (PAK2) Serine/threonine-protein kinase pak 2 (PAK2)
15丝氨酸/苏氨酸蛋白激酶 stk11 (STK11) Serine/threonine-protein kinase stk11 (STK11)
2受体相互作用丝氨酸/苏氨酸蛋白激酶3 (RIPK3) Receptor-interacting serine/threonine-protein kinase 3 (RIPK3)
395'-AMP激活蛋白激酶亚基γ-1 (PRKAG1) 5'-AMP-activated protein kinase subunit gamma-1 (PRKAG1)
38丝裂原活化蛋白激酶激酶激酶 6 (MAP3K6) Mitogen-activated protein kinase kinase kinase 6 (MAP3K6)
4成纤维细胞生长因子受体3(FGFR3) Fibroblast growth factor receptor 3 (FGFR3)
64肌球蛋白轻链激酶3 (MYLK3) Myosin light chain kinase 3 (MYLK3)
5Ephrin a 型受体 1 (EPHA1) Ephrin type-a receptor 1 (EPHA1)
12丝氨酸/苏氨酸蛋白激酶 ICK (ICK) Serine/threonine-protein kinase ick (ICK)
0酪氨酸蛋白激酶受体ufo(AXL) Tyrosine-protein kinase receptor ufo (AXL)
98腺苷激酶(ADK) Adenosine kinase (ADK)
26双特异性睾丸特异性蛋白激酶1 (TESK1) Dual specificity testis-specific protein kinase 1 (TESK1)
6酪氨酸蛋白激酶 itk/tsk (ITK) Tyrosine-protein kinase itk/tsk (ITK)
34细胞周期蛋白依赖性激酶17 (CDK17) Cyclin-dependent kinase 17 (CDK17)
6Ephrin a 型受体 7 (EPHA7) Ephrin type-a receptor 7 (EPHA7)
1脱氧胞苷激酶(DCK) Deoxycytidine kinase (DCK)
7丝氨酸/苏氨酸蛋白激酶 mrck gamma (CDC42BPG) Serine/threonine-protein kinase mrck gamma (CDC42BPG)
2死亡相关蛋白激酶3 (DAPK3) Death-associated protein kinase 3 (DAPK3)
11吡哆醛激酶(PDXK) Pyridoxal kinase (PDXK)
2Tp53调节激酶(TP53RK) Tp53-regulating kinase (TP53RK)
0未表征的含Aarf结构域的蛋白激酶1(ADCK1) Uncharacterized aarf domain-containing protein kinase 1 (ADCK1)
2丝氨酸/苏氨酸蛋白激酶α-raf(ARAF) Serine/threonine-protein kinase a-raf (ARAF)
7丝氨酸/苏氨酸蛋白激酶 plk3 (PLK3) Serine/threonine-protein kinase plk3 (PLK3)
21丝氨酸/苏氨酸蛋白激酶/核糖核酸内切酶ire2 (ERN2) Serine/threonine-protein kinase/endoribonuclease ire2 (ERN2)
0线粒体腺苷酸激酶2 (AK2) Adenylate kinase 2, mitochondrial (AK2)
0受体酪氨酸蛋白激酶 erbb-4 (ERBB4) Receptor tyrosine-protein kinase erbb-4 (ERBB4)
52富含亮氨酸重复丝氨酸/苏氨酸蛋白激酶 2 (LRRK2) Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)
99Map激酶相互作用丝氨酸/苏氨酸蛋白激酶2 (MKNK2) Map kinase-interacting serine/threonine-protein kinase 2 (MKNK2)
52Ste20相关激酶衔接蛋白α(STRADA) Ste20-related kinase adapter protein alpha (STRADA)
2酪氨酸蛋白激酶受体 tyro3 (TYRO3) Tyrosine-protein kinase receptor tyro3 (TYRO3)
24双特异性蛋白激酶 TTK (TTK) Dual specificity protein kinase ttk (TTK)
49Nt-3生长因子受体(NTRK3) Nt-3 growth factor receptor (NTRK3)
51有丝分裂检查点丝氨酸/苏氨酸蛋白激酶 bub1 (BUB1) Mitotic checkpoint serine/threonine-protein kinase bub1 (BUB1)
8丝氨酸/苏氨酸蛋白激酶24 (STK24) Serine/threonine-protein kinase 24 (STK24)
5整合素连接蛋白激酶(ILK) Integrin-linked protein kinase (ILK)
5双特异性蛋白激酶 clk3 (CLK3) Dual specificity protein kinase clk3 (CLK3)
17丝氨酸/苏氨酸蛋白激酶 PAK 1 (PAK1) Serine/threonine-protein kinase pak 1 (PAK1)
30MAP激酶激活蛋白激酶3 (MAPKAPK3) Map kinase-activated protein kinase 3 (MAPKAPK3)
4酪氨酸蛋白激酶 BLK Tyrosine-protein kinase blk (BLK)
40丝氨酸/苏氨酸蛋白激酶 chk2 (CHEK2) Serine/threonine-protein kinase chk2 (CHEK2)
20ATP依赖性6-磷酸果糖激酶,血小板型(PFKP) ATP-dependent 6-phosphofructokinase, platelet type (PFKP)
2丝裂原活化蛋白激酶 12 (MAPK12) Mitogen-activated protein kinase 12 (MAPK12)
8丝氨酸/苏氨酸蛋白激酶 pim-3 (PIM3) Serine/threonine-protein kinase pim-3 (PIM3)
42磷脂酰肌醇 5-磷酸 4-激酶 2 型 α (PIP4K2A) Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha (PIP4K2A)
15依赖营地的蛋白激酶催化亚基prkx(PRKX) Camp-dependent protein kinase catalytic subunit prkx (PRKX)
4细胞周期蛋白依赖性激酶 8 (CDK8) Cyclin-dependent kinase 8 (CDK8)
52丝裂原活化蛋白激酶13 (MAPK13) Mitogen-activated protein kinase 13 (MAPK13)
9丝氨酸/苏氨酸蛋白激酶 PAK 6 (PAK6) Serine/threonine-protein kinase pak 6 (PAK6)
5钙/钙调蛋白依赖性蛋白激酶1型(CAMK1) Calcium/calmodulin-dependent protein kinase type 1 (CAMK1)
0核因子 kappa-b 激酶亚基 α 抑制剂 (CHUK) Inhibitor of nuclear factor kappa-b kinase subunit alpha (CHUK)
42依赖营地的蛋白激酶催化亚基γ (PRKACG) Camp-dependent protein kinase catalytic subunit gamma (PRKACG)
3细胞周期蛋白依赖性激酶样蛋白5 (CDKL5) Cyclin-dependent kinase-like 5 (CDKL5)
12含PAS结构域的丝氨酸/苏氨酸蛋白激酶(PASK) Pas domain-containing serine/threonine-protein kinase (PASK)
4酪氨酸蛋白激酶聚合体 (MERTK) Tyrosine-protein kinase mer (MERTK)
41丝氨酸/苏氨酸蛋白激酶 nek7 (NEK7) Serine/threonine-protein kinase nek7 (NEK7)
5Srsf蛋白激酶1(SRPK1) Srsf protein kinase 1 (SRPK1)
15血管生成素-1受体(TEK) Angiopoietin-1 receptor (TEK)
39同源域相互作用蛋白激酶2 (HIPK2) Homeodomain-interacting protein kinase 2 (HIPK2)
12丝氨酸/苏氨酸蛋白激酶 dclk1 (DCLK1) Serine/threonine-protein kinase dclk1 (DCLK1)
12丝氨酸/苏氨酸蛋白激酶brsk1(BRSK1) Serine/threonine-protein kinase brsk1 (BRSK1)
1G蛋白偶联受体激酶6(GRK6) G protein-coupled receptor kinase 6 (GRK6)
11丝氨酸/苏氨酸蛋白激酶17a (STK17A) Serine/threonine-protein kinase 17a (STK17A)
21钙/钙调蛋白依赖性蛋白激酶II型β亚基(CAMK2B) Calcium/calmodulin-dependent protein kinase type ii subunit beta (CAMK2B)
1原癌基因酪氨酸蛋白激酶 ros (ROS1) Proto-oncogene tyrosine-protein kinase ros (ROS1)
39钙/钙调蛋白依赖性蛋白激酶II型亚基α(CAMK2A) Calcium/calmodulin-dependent protein kinase type ii subunit alpha (CAMK2A)
30Raf原癌基因丝氨酸/苏氨酸蛋白激酶(RAF1) Raf proto-oncogene serine/threonine-protein kinase (RAF1)
79同源域相互作用蛋白激酶 4 (HIPK4) Homeodomain-interacting protein kinase 4 (HIPK4)
6白细胞酪氨酸激酶受体(LTK) Leukocyte tyrosine kinase receptor (LTK)
12蛋白激酶cγ型(PRKCG) Protein kinase c gamma type (PRKCG)
12推测的己糖激酶 HKDC1 (HKDC1) Putative hexokinase HKDC1 (HKDC1)
27丝氨酸/苏氨酸蛋白激酶 nek4 (NEK4) Serine/threonine-protein kinase nek4 (NEK4)
0睾丸特异性丝氨酸/苏氨酸蛋白激酶 1 (TSSK1B) Testis-specific serine/threonine-protein kinase 1 (TSSK1B)
1钙/钙调蛋白依赖性蛋白激酶1d型(CAMK1D) Calcium/calmodulin-dependent protein kinase type 1d (CAMK1D)
3双特异性丝裂原活化蛋白激酶激酶 4 (MAP2K4) Dual specificity mitogen-activated protein kinase kinase 4 (MAP2K4)
10Cgmp依赖性蛋白激酶2(PRKG2) Cgmp-dependent protein kinase 2 (PRKG2)
1丝氨酸/苏氨酸蛋白激酶38样蛋白(STK38L) Serine/threonine-protein kinase 38-like (STK38L)
0丝氨酸/苏氨酸蛋白激酶ATR(ATR) Serine/threonine-protein kinase atr (ATR)
37酪氨酸蛋白激酶 fgr (FGR) Tyrosine-protein kinase fgr (FGR)
13成纤维细胞生长因子受体2(FGFR2) Fibroblast growth factor receptor 2 (FGFR2)
74Map激酶相互作用丝氨酸/苏氨酸蛋白激酶1 (MKNK1) Map kinase-interacting serine/threonine-protein kinase 1 (MKNK1)
49酪氨酸蛋白激酶 srms (SRMS) Tyrosine-protein kinase srms (SRMS)
6酪氨酸蛋白激酶 ZAP-70 (ZAP70) Tyrosine-protein kinase zap-70 (ZAP70)
14巨核细胞相关酪氨酸蛋白激酶(MATK) Megakaryocyte-associated tyrosine-protein kinase (MATK)
0丝氨酸/苏氨酸蛋白激酶 SGK2 (SGK2) Serine/threonine-protein kinase sgk2 (SGK2)
4双特异性睾丸特异性蛋白激酶2 (TESK2) Dual specificity testis-specific protein kinase 2 (TESK2)
6丝氨酸/苏氨酸蛋白激酶n3(PKN3) Serine/threonine-protein kinase n3 (PKN3)
1双特异性酪氨酸磷酸化调节激酶3 (DYRK3) Dual specificity tyrosine-phosphorylation-regulated kinase 3 (DYRK3)
8未表征的含Aarf结构域的蛋白激酶5(ADCK5) Uncharacterized aarf domain-containing protein kinase 5 (ADCK5)
0丝氨酸/苏氨酸蛋白激酶38 (STK38) Serine/threonine-protein kinase 38 (STK38)
0细胞质酪氨酸蛋白激酶 BMX (BMX) Cytoplasmic tyrosine-protein kinase bmx (BMX)
53成纤维细胞生长因子受体 4 (FGFR4) Fibroblast growth factor receptor 4 (FGFR4)
62受体相互作用丝氨酸/苏氨酸蛋白激酶 1 (RIPK1) Receptor-interacting serine/threonine-protein kinase 1 (RIPK1)
71细胞周期蛋白依赖性激酶19 (CDK19) Cyclin-dependent kinase 19 (CDK19)
18双特异性酪氨酸磷酸化调节激酶2 (DYRK2) Dual specificity tyrosine-phosphorylation-regulated kinase 2 (DYRK2)
28磷脂酰肌醇4-激酶β(PI4KB) Phosphatidylinositol 4-kinase beta (PI4KB)
35蛋白激酶cε型(PRKCE) Protein kinase c epsilon type (PRKCE)
36UMP-CMP激酶(CMPK1) UMP-CMP kinase (CMPK1)
2G蛋白偶联受体激酶5(GRK5) G protein-coupled receptor kinase 5 (GRK5)
13双特异性酪氨酸磷酸化调节激酶 4 (DYRK4) Dual specificity tyrosine-phosphorylation-regulated kinase 4 (DYRK4)
0丝氨酸/苏氨酸蛋白激酶受体 r3 (ACVRL1) Serine/threonine-protein kinase receptor r3 (ACVRL1)
23DNA依赖性蛋白激酶催化亚基(PRKDC) Dna-dependent protein kinase catalytic subunit (PRKDC)
97丝裂原活化蛋白激酶激酶激酶9 (MAP3K9) Mitogen-activated protein kinase kinase kinase 9 (MAP3K9)
125'-AMP激活蛋白激酶催化亚基α-2 (PRKAA2) 5'-AMP-activated protein kinase catalytic subunit alpha-2 (PRKAA2)
37干扰素诱导的双链RNA激活蛋白激酶(EIF2AK2) Interferon-induced, double-stranded rna-activated protein kinase (EIF2AK2)
30死亡相关蛋白激酶 1 (DAPK1) Death-associated protein kinase 1 (DAPK1)
17丝氨酸/苏氨酸蛋白激酶d1(PRKD1) Serine/threonine-protein kinase d1 (PRKD1)
23Nuak家族snf1样激酶1(NUAK1) Nuak family snf1-like kinase 1 (NUAK1)
19淋巴因子激活的杀伤性T细胞来源蛋白激酶(PBK) Lymphokine-activated killer t-cell-originated protein kinase (PBK)
1酪氨酸蛋白激酶 TXK (TXK) Tyrosine-protein kinase txk (TXK)
19极光激酶c(AURKC) Aurora kinase c (AURKC)
25丝裂原活化蛋白激酶激酶激酶10 (MAP3K10) Mitogen-activated protein kinase kinase kinase 10 (MAP3K10)
1磷脂酰肌醇 4-磷酸 3-激酶 c2 结构域亚基 β (PIK3C2B) Phosphatidylinositol 4-phosphate 3-kinase c2 domain-containing subunit beta (PIK3C2B)
24核糖体蛋白S6激酶α-2(RPS6KA2) Ribosomal protein s6 kinase alpha-2 (RPS6KA2)
20丝氨酸/苏氨酸蛋白激酶 nek6 (NEK6) Serine/threonine-protein kinase nek6 (NEK6)
4丝裂原活化蛋白激酶激酶激酶7 (MAP3K7) Mitogen-activated protein kinase kinase kinase 7 (MAP3K7)
29睾丸特异性丝氨酸/苏氨酸蛋白激酶2 (TSSK2) Testis-specific serine/threonine-protein kinase 2 (TSSK2)
1蛋白激酶c eta型(PRKCH) Protein kinase c eta type (PRKCH)
13钙/钙调蛋白依赖性蛋白激酶1g型(CAMK1G) Calcium/calmodulin-dependent protein kinase type 1g (CAMK1G)
4细胞周期蛋白依赖性激酶18 (CDK18) Cyclin-dependent kinase 18 (CDK18)
0Ephrin a 型受体 3 (EPHA3) Ephrin type-a receptor 3 (EPHA3)
14真核延伸因子2激酶(EEF2K) Eukaryotic elongation factor 2 kinase (EEF2K)
10Ephrin B 型受体 1 (EPHB1) Ephrin type-b receptor 1 (EPHB1)
2双特异性丝裂原活化蛋白激酶激酶7 (MAP2K7) Dual specificity mitogen-activated protein kinase kinase 7 (MAP2K7)
11肌肉骨骼受体酪氨酸蛋白激酶(MUSK) Muscle, skeletal receptor tyrosine-protein kinase (MUSK)
2丝氨酸/苏氨酸蛋白激酶mark1(MARK1) Serine/threonine-protein kinase mark1 (MARK1)
4丝氨酸/苏氨酸蛋白激酶 PAK 3 (PAK3) Serine/threonine-protein kinase pak 3 (PAK3)
8真核翻译起始因子2-α激酶3 (EIF2AK3) Eukaryotic translation initiation factor 2-alpha kinase 3 (EIF2AK3)
26丝氨酸/苏氨酸蛋白激酶33 (STK33) Serine/threonine-protein kinase 33 (STK33)
4丝氨酸/苏氨酸蛋白激酶 tousled-like 2 (TLK2) Serine/threonine-protein kinase tousled-like 2 (TLK2)
10Ephrin a 型受体 8 (EPHA8) Ephrin type-a receptor 8 (EPHA8)
4丝氨酸/苏氨酸蛋白激酶 sik1 (SIK1) Serine/threonine-protein kinase sik1 (SIK1)
9Ephrin a 型受体 6 (EPHA6) Ephrin type-a receptor 6 (EPHA6)
1丝氨酸/苏氨酸蛋白激酶 plk2 (PLK2) Serine/threonine-protein kinase plk2 (PLK2)
12Srsf蛋白激酶2(SRPK2) Srsf protein kinase 2 (SRPK2)
10真核翻译起始因子2α激酶4(EIF2AK4) Eukaryotic translation initiation factor 2-alpha kinase 4 (EIF2AK4)
13同源域相互作用蛋白激酶1 (HIPK1) Homeodomain-interacting protein kinase 1 (HIPK1)
4丝氨酸/苏氨酸蛋白激酶 brsk2 (BRSK2) Serine/threonine-protein kinase brsk2 (BRSK2)
4丝氨酸/苏氨酸蛋白激酶 dclk2 (DCLK2) Serine/threonine-protein kinase dclk2 (DCLK2)
4丝氨酸/苏氨酸蛋白激酶 PAK7 (PAK7) Serine/threonine-protein kinase pak 7 (PAK7)
6胰岛素受体相关蛋白(INSRR) Insulin receptor-related protein (INSRR)
2丝氨酸/苏氨酸蛋白激酶17b (STK17B) Serine/threonine-protein kinase 17b (STK17B)
11钙/钙调蛋白依赖性蛋白激酶激酶1 (CAMKK1) Calcium/calmodulin-dependent protein kinase kinase 1 (CAMKK1)
6细胞周期蛋白依赖性激酶11b (CDK11B) Cyclin-dependent kinase 11b (CDK11B)
4丝裂原活化蛋白激酶 6 (MAPK6) Mitogen-activated protein kinase 6 (MAPK6)
4肌球蛋白轻链激酶2,骨骼肌/心肌(MYLK2) Myosin light chain kinase 2, skeletal/cardiac muscle (MYLK2)
0肌强直蛋白激酶 (DMPK) Myotonin-protein kinase (DMPK)
1丝氨酸/苏氨酸蛋白激酶 ULK2 (ULK2) Serine/threonine-protein kinase ulk2 (ULK2)
9磷脂酰肌醇 5-磷酸 4-激酶 2 型 β (PIP4K2B) Phosphatidylinositol 5-phosphate 4-kinase type-2 beta (PIP4K2B)
8磷酸化酶b激酶γ催化链,骨骼肌/心肌同工型(PHKG1) Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform (PHKG1)
3受体酪氨酸蛋白激酶 erbb-3 (ERBB3) Receptor tyrosine-protein kinase erbb-3 (ERBB3)
19丝氨酸/苏氨酸蛋白激酶25 (STK25) Serine/threonine-protein kinase 25 (STK25)
0丝氨酸/苏氨酸蛋白激酶 tnni3k (TNNI3K) Serine/threonine-protein kinase tnni3k (TNNI3K)
5酪氨酸蛋白激酶受体 Tie-1 (TIE1) Tyrosine-protein kinase receptor tie-1 (TIE1)
7死亡相关蛋白激酶 2 (DAPK2) Death-associated protein kinase 2 (DAPK2)
2肌球蛋白轻链激酶家族成员4(MYLK4) Myosin light chain kinase family member 4 (MYLK4)
5磷脂酰肌醇 4-磷酸 5-激酶 1 型 α (PIP5K1A) Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha (PIP5K1A)
0视紫红质激酶(GRK1) Rhodopsin kinase (GRK1)
9丝氨酸/苏氨酸蛋白激酶 nim1 (NIM1K) Serine/threonine-protein kinase nim1 (NIM1K)
0丝裂原活化蛋白激酶 4 (MAPK4) Mitogen-activated protein kinase 4 (MAPK4)
0丝氨酸/苏氨酸蛋白激酶 lats2 (LATS2) Serine/threonine-protein kinase lats2 (LATS2)
2丝氨酸/苏氨酸蛋白激酶 tousled-like 1 (TLK1) Serine/threonine-protein kinase tousled-like 1 (TLK1)
0Srsf蛋白激酶3(SRPK3) Srsf protein kinase 3 (SRPK3)
8激活素受体2a型(ACVR2A) Activin receptor type-2a (ACVR2A)
4细胞周期蛋白依赖性激酶11a (CDK11A) Cyclin-dependent kinase 11a (CDK11A)
4细胞周期蛋白依赖性激酶14 (CDK14) Cyclin-dependent kinase 14 (CDK14)
4丝裂原活化蛋白激酶激酶激酶19 (MAP3K19) Mitogen-activated protein kinase kinase kinase 19 (MAP3K19)
13肌球蛋白-iiib (MYO3B) Myosin-iiib (MYO3B)
0磷脂酰肌醇 4-磷酸 3-激酶 c2 结构域亚基 γ (PIK3C2G) Phosphatidylinositol 4-phosphate 3-kinase c2 domain-containing subunit gamma (PIK3C2G)
8丝氨酸/苏氨酸蛋白激酶 32c (STK32C) Serine/threonine-protein kinase 32c (STK32C)
1丝氨酸/苏氨酸蛋白激酶36 (STK36) Serine/threonine-protein kinase 36 (STK36)
0丝氨酸/苏氨酸蛋白激酶 dclk3 (DCLK3) Serine/threonine-protein kinase dclk3 (DCLK3)
5丝氨酸/苏氨酸蛋白激酶 rio1 (RIOK1) Serine/threonine-protein kinase rio1 (RIOK1)
2丝氨酸/苏氨酸蛋白激酶 rio3 (RIOK3) Serine/threonine-protein kinase rio3 (RIOK3)
0丝氨酸/苏氨酸蛋白激酶 SGK3 (SGK3) Serine/threonine-protein kinase sgk3 (SGK3)
5含Aarf结构域的蛋白激酶4(ADCK4) Aarf domain-containing protein kinase 4 (ADCK4)
0同源域相互作用蛋白激酶3 (HIPK3) Homeodomain-interacting protein kinase 3 (HIPK3)
0丝氨酸/苏氨酸蛋白激酶32b (STK32B) Serine/threonine-protein kinase 32b (STK32B)
0丝氨酸/苏氨酸蛋白激酶 nek5 (NEK5) Serine/threonine-protein kinase nek5 (NEK5)
2锚蛋白重复序列和蛋白激酶结构域蛋白1 (ANKK1) Ankyrin repeat and protein kinase domain-containing protein 1 (ANKK1)
0酪蛋白激酶 I 同工型 α 样 (CSNK1A1L) Casein kinase i isoform alpha-like (CSNK1A1L)
0G蛋白偶联受体激酶7(GRK7) G protein-coupled receptor kinase 7 (GRK7)
0肌球蛋白-IIIa (MYO3A) Myosin-iiia (MYO3A)
0磷脂酰肌醇 4-磷酸 5-激酶 1 型 γ (PIP5K1C) Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma (PIP5K1C)
7Wee1样蛋白激酶2(WEE2) Wee1-like protein kinase 2 (WEE2)
3细胞周期蛋白依赖性激酶样蛋白2 (CDKL2) Cyclin-dependent kinase-like 2 (CDKL2)
10磷脂酰肌醇3-激酶调节亚基α(PIK3R1) Phosphatidylinositol 3-kinase regulatory subunit alpha (PIK3R1)
96G蛋白偶联受体激酶4(GRK4) G protein-coupled receptor kinase 4 (GRK4)
0丝氨酸/苏氨酸蛋白激酶 rio2 (RIOK2) Serine/threonine-protein kinase rio2 (RIOK2)
4受体相互作用丝氨酸/苏氨酸蛋白激酶 4 (RIPK4) Receptor-interacting serine/threonine-protein kinase 4 (RIPK4)
0丝氨酸/苏氨酸蛋白激酶 vrk2 (VRK2) Serine/threonine-protein kinase vrk2 (VRK2)
2Ste20/sps1 相关富含脯氨酸-丙氨酸的蛋白激酶 (STK39) Ste20/sps1-related proline-alanine-rich protein kinase (STK39)
0细胞周期蛋白依赖性激酶样蛋白3 (CDKL3) Cyclin-dependent kinase-like 3 (CDKL3)
3双丝氨酸/苏氨酸和酪氨酸蛋白激酶(DSTYK) Dual serine/threonine and tyrosine protein kinase (DSTYK)
0丝裂原活化蛋白激酶激酶激酶12 (MAP3K12) Mitogen-activated protein kinase kinase kinase 12 (MAP3K12)
5丝裂原活化蛋白激酶激酶激酶13 (MAP3K13) Mitogen-activated protein kinase kinase kinase 13 (MAP3K13)
4丝氨酸/苏氨酸蛋白激酶 nek11 (NEK11) Serine/threonine-protein kinase nek11 (NEK11)
0细胞周期蛋白依赖性激酶15 (CDK15) Cyclin-dependent kinase 15 (CDK15)
0半乳糖激酶(GALK1) Galactokinase (GALK1)
25丝氨酸/苏氨酸蛋白激酶prp4同源物(PRPF4B) Serine/threonine-protein kinase prp4 homolog (PRPF4B)
0激素上调的神经肿瘤相关激酶(HUNK) Hormonally up-regulated neu tumor-associated kinase (HUNK)
0微管相关丝氨酸/苏氨酸蛋白激酶1 (MAST1) Microtubule-associated serine/threonine-protein kinase 1 (MAST1)
0丝裂原活化蛋白激酶激酶激酶15 (MAP3K15) Mitogen-activated protein kinase kinase kinase 15 (MAP3K15)
0丝氨酸/苏氨酸蛋白激酶35 (STK35) Serine/threonine-protein kinase 35 (STK35)
2丝氨酸/苏氨酸蛋白激酶 MAK (MAK) Serine/threonine-protein kinase mak (MAK)
0丝氨酸/苏氨酸蛋白激酶 osr1 (OXSR1) Serine/threonine-protein kinase osr1 (OXSR1)
0未表征的丝氨酸/苏氨酸蛋白激酶 sbk3 (SBK3) Uncharacterized serine/threonine-protein kinase sbk3 (SBK3)
0细胞周期蛋白依赖性激酶样蛋白1 (CDKL1) Cyclin-dependent kinase-like 1 (CDKL1)
1外周质膜蛋白 cask (CASK) Peripheral plasma membrane protein cask (CASK)
0磷脂酰肌醇3-激酶催化亚基3型(PIK3C3) Phosphatidylinositol 3-kinase catalytic subunit type 3 (PIK3C3)
48丝氨酸/苏氨酸蛋白激酶32a (STK32A) Serine/threonine-protein kinase 32a (STK32A)
0丝氨酸/苏氨酸蛋白激酶 sbk1 (SBK1) Serine/threonine-protein kinase sbk1 (SBK1)
0Snf相关丝氨酸/苏氨酸蛋白激酶(SNRK) Snf-related serine/threonine-protein kinase (SNRK)
0瞬时受体电位阳离子通道亚家族m成员6(TRPM6) Transient receptor potential cation channel subfamily m member 6 (TRPM6)
2[丙酮酸脱氢酶(乙酰转移)]激酶同工酶1,线粒体(PDK1) [pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial (PDK1)
31细胞周期蛋白依赖性激酶10 (CDK10) Cyclin-dependent kinase 10 (CDK10)
0己糖激酶-1 (HK1) Hexokinase-1 (HK1)
7丝氨酸/苏氨酸蛋白激酶 SGK1 (SGK1) Serine/threonine-protein kinase sgk1 (SGK1)
12丝裂原活化蛋白激酶激酶激酶14 (MAP3K14) Mitogen-activated protein kinase kinase kinase 14 (MAP3K14)
225'-AMP激活蛋白激酶亚基β-1(PRKAB1) 5'-AMP-activated protein kinase subunit beta-1 (PRKAB1)
32酪蛋白激酶 II β 亚基 (CSNK2B) Casein kinase ii subunit beta (CSNK2B)
27鞘氨醇激酶1(SPHK1) Sphingosine kinase 1 (SPHK1)
35转录起始因子 tfiid 亚基 1 (TAF1) Transcription initiation factor tfiid subunit 1 (TAF1)
48葡萄糖激酶(GCK) Glucokinase (GCK)
30丝氨酸/苏氨酸蛋白激酶 haspin (GSG2) Serine/threonine-protein kinase haspin (GSG2)
17磷脂酰肌醇4-激酶α(PI4KA) Phosphatidylinositol 4-kinase alpha (PI4KA)
14鞘氨醇激酶 2 (SPHK2) Sphingosine kinase 2 (SPHK2)
29胞质胸苷激酶(TK1) Thymidine kinase, cytosolic (TK1)
30丝裂原活化蛋白激酶激酶激酶 8 (MAP3K8) Mitogen-activated protein kinase kinase kinase 8 (MAP3K8)
7肌醇六磷酸激酶 2 (IP6K2) Inositol hexakisphosphate kinase 2 (IP6K2)
28含磷脂酰肌醇 4-磷酸 3-激酶 c2 结构域的亚基 α (PIK3C2A) Phosphatidylinositol 4-phosphate 3-kinase c2 domain-containing subunit alpha (PIK3C2A)
8肌醇多磷酸多激酶(IPMK) Inositol polyphosphate multikinase (IPMK)
26[丙酮酸脱氢酶(乙酰转移)]激酶同工酶2,线粒体(PDK2) [pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial (PDK2)
24核苷二磷酸激酶B(NME1-NME2) Nucleoside diphosphate kinase B (NME1-NME2)
2丙酮酸激酶 PKLR (PKLR) Pyruvate kinase PKLR (PKLR)
176-磷酸果糖-2-激酶/果糖-2,6-二磷酸酶 3 (PFKFB3) 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3 (PFKFB3)
17丝氨酸/苏氨酸蛋白激酶 WNK1 (WNK1) Serine/threonine-protein kinase wnk1 (WNK1)
5[丙酮酸脱氢酶(乙酰转移)]激酶同工酶4,线粒体(PDK4) [pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial (PDK4)
221-磷脂酰肌醇3-磷酸5-激酶(PIKFYVE) 1-phosphatidylinositol 3-phosphate 5-kinase (PIKFYVE)
14胆碱激酶α(CHKA) Choline kinase alpha (CHKA)
10丝氨酸/苏氨酸蛋白激酶 WNK2 (WNK2) Serine/threonine-protein kinase wnk2 (WNK2)
0二酰甘油激酶α (DGKA) Diacylglycerol kinase alpha (DGKA)
14β-肾上腺素能受体激酶2 (ADRBK2) Beta-adrenergic receptor kinase 2 (ADRBK2)
4Nf-kappa-b 必需调节因子 (IKBKG) Nf-kappa-b essential modulator (IKBKG)
6推测的核苷二磷酸激酶(NME2P1) Putative nucleoside diphosphate kinase (NME2P1)
0核糖体蛋白S6激酶β-2(RPS6KB2) Ribosomal protein s6 kinase beta-2 (RPS6KB2)
1[丙酮酸脱氢酶(乙酰转移)]激酶同工酶3,线粒体(PDK3) [pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial (PDK3)
162-5a依赖性核糖核酸酶(RNASEL) 2-5a-dependent ribonuclease (RNASEL)
11钙/钙调蛋白依赖性蛋白激酶1b型(PNCK) Calcium/calmodulin-dependent protein kinase type 1b (PNCK)
1肌醇六磷酸激酶 1 (IP6K1) Inositol hexakisphosphate kinase 1 (IP6K1)
2丝氨酸/苏氨酸蛋白激酶 vrk1 (VRK1) Serine/threonine-protein kinase vrk1 (VRK1)
2丝氨酸/苏氨酸蛋白激酶 WNK3 (WNK3) Serine/threonine-protein kinase wnk3 (WNK3)
0TGF-β激活激酶1和MAP3K7结合蛋白1(TAB1) Tgf-beta-activated kinase 1 and map3k7-binding protein 1 (TAB1)
2线粒体胸苷激酶2 (TK2) Thymidine kinase 2, mitochondrial (TK2)
5肌醇六磷酸激酶 3 (IP6K3) Inositol hexakisphosphate kinase 3 (IP6K3)
2酮己糖激酶(KHK) Ketohexokinase (KHK)
7混合谱系激酶结构域样蛋白(MLKL) Mixed lineage kinase domain-like protein (MLKL)
4丝氨酸/苏氨酸蛋白激酶lmtk3 (LMTK3) Serine/threonine-protein kinase lmtk3 (LMTK3)
2丝氨酸/苏氨酸蛋白激酶 smg1 (SMG1) Serine/threonine-protein kinase smg1 (SMG1)
9Tau蛋白-微管蛋白激酶1(TTBK1) Tau-tubulin kinase 1 (TTBK1)
3睾丸特异性丝氨酸/苏氨酸蛋白激酶3 (TSSK3) Testis-specific serine/threonine-protein kinase 3 (TSSK3)
0胸苷酸激酶(DTYMK) Thymidylate kinase (DTYMK)
9心房利钠肽受体 1 (NPR1) Atrial natriuretic peptide receptor 1 (NPR1)
5泛酸激酶3 (PANK3) Pantothenate kinase 3 (PANK3)
3磷脂酰肌醇 4-激酶 2-α 型 (PI4K2A) Phosphatidylinositol 4-kinase type 2-alpha (PI4K2A)
1丝氨酸/苏氨酸蛋白激酶 nek10 (NEK10) Serine/threonine-protein kinase nek10 (NEK10)
3甘油激酶(GK) Glycerol kinase (GK)
2NAD激酶(NADK) NAD kinase (NADK)
4磷酸甘油酸激酶1(PGK1) Phosphoglycerate kinase 1 (PGK1)
1Tau蛋白-微管蛋白激酶2 (TTBK2) Tau-tubulin kinase 2 (TTBK2)
1尿苷胞苷激酶2 (UCK2) Uridine-cytidine kinase 2 (UCK2)
06-磷酸果糖-2-激酶/果糖-2,6-二磷酸酶 1 (PFKFB1) 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 1 (PFKFB1)
36-磷酸果糖-2-激酶/果糖-2,6-二磷酸酶 2 (PFKFB2) 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 2 (PFKFB2)
3细胞周期蛋白依赖性激酶 20 (CDK20) Cyclin-dependent kinase 20 (CDK20)
0己糖激酶-2 (HK2) Hexokinase-2 (HK2)
4酮胺-3-激酶(FN3KRP) Ketosamine-3-kinase (FN3KRP)
0核糖磷酸焦磷酸激酶1 (PRPS1) Ribose-phosphate pyrophosphokinase 1 (PRPS1)
2丝氨酸/苏氨酸蛋白激酶 nek8 (NEK8) Serine/threonine-protein kinase nek8 (NEK8)
0睾丸特异性丝氨酸/苏氨酸蛋白激酶 6 (TSSK6) Testis-specific serine/threonine-protein kinase 6 (TSSK6)
0ATP依赖性6-磷酸果糖激酶,肝型(PFKL) Atp-dependent 6-phosphofructokinase, liver type (PFKL)
0细胞周期蛋白依赖性激酶样蛋白4 (CDKL4) Cyclin-dependent kinase-like 4 (CDKL4)
3果糖胺-3-激酶(FN3K) Fructosamine-3-kinase (FN3K)
0白细胞介素-1受体相关激酶样2(IRAK2) Interleukin-1 receptor-associated kinase-like 2 (IRAK2)
0ras 1 激酶抑制因子 (KSR1) Kinase suppressor of ras 1 (KSR1)
0Ras 2 激酶抑制因子 (KSR2) Kinase suppressor of ras 2 (KSR2)
0微管相关丝氨酸/苏氨酸蛋白激酶3 (MAST3) Microtubule-associated serine/threonine-protein kinase 3 (MAST3)
0丝裂原活化蛋白激酶激酶激酶 mlk4 (MLK4) Mitogen-activated protein kinase kinase kinase mlk4 (MLK4)
0核苷二磷酸激酶A(NME1) Nucleoside diphosphate kinase A (NME1)
0Pab依赖性多聚腺苷酸特异性核糖核酸酶亚基pan3(PAN3) Pab-dependent poly(a)-specific ribonuclease subunit pan3 (PAN3)
0泛酸激酶1 (PANK1) Pantothenate kinase 1 (PANK1)
1线粒体泛酸激酶2 (PANK2) Pantothenate kinase 2, mitochondrial (PANK2)
1磷酸烯醇式丙酮酸羧激酶 [gtp],线粒体 (PCK2) Phosphoenolpyruvate carboxykinase [gtp], mitochondrial (PCK2)
0胞质磷酸烯醇式丙酮酸羧激酶[GTP] (PCK1) Phosphoenolpyruvate carboxykinase, cytosolic [GTP] (PCK1)
1磷脂酰肌醇3-激酶调节亚基4(PIK3R4) Phosphoinositide 3-kinase regulatory subunit 4 (PIK3R4)
2磷酸化酶b激酶调节亚基α,肝脏同工型(PHKA2) Phosphorylase b kinase regulatory subunit alpha, liver isoform (PHKA2)
0伪足富集非典型激酶 1 (PEAK1) Pseudopodium-enriched atypical kinase 1 (PEAK1)
0丝氨酸/苏氨酸蛋白激酶31 (STK31) Serine/threonine-protein kinase 31 (STK31)
0丝氨酸/苏氨酸蛋白激酶长城(MASTL) Serine/threonine-protein kinase greatwall (MASTL)
0丝氨酸/苏氨酸蛋白激酶lmtk2 (LMTK2) Serine/threonine-protein kinase lmtk2 (LMTK2)
0丝氨酸/苏氨酸蛋白激酶 WNK4 (WNK4) Serine/threonine-protein kinase wnk4 (WNK4)
0Ste20相关激酶衔接蛋白β(STRADB) Ste20-related kinase adapter protein beta (STRADB)
0肌联蛋白(TTN) Titin (TTN)
0三功能域蛋白(TRIO) Triple functional domain protein (TRIO)
2产品列表
-
甲氧滴滴涕分析标准品 ? 分析标准品 —— 纯度认证的材料,供定量校准使用。用于配制校准标准并验证分析方法。有现货 货号: M114227查看产品价格与包装
技术标识符
- IUPAC名称
- 1-methoxy-4-[2,2,2-trichloro-1-(4-methoxyphenyl)ethyl]benzene
- SMILES
- COC1=CC=C(C=C1)C(C2=CC=C(C=C2)OC)C(Cl)(Cl)Cl
- InChIKey
- IAKOZHOLGAGEJT-UHFFFAOYSA-N
- InChI
- 1S/C16H15Cl3O2/c1-20-13-7-3-11(4-8-13)15(16(17,18)19)12-5-9-14(21-2)10-6-12/h3-10,15H,1-2H3
-
2-溴-4'-甲基苯乙酮有现货 货号: M113665查看产品价格与包装
技术标识符
- IUPAC名称
- 2-bromo-1-(4-methylphenyl)ethanone
- SMILES
- CC1=CC=C(C=C1)C(=O)CBr
- InChIKey
- KRVGXFREOJHJAX-UHFFFAOYSA-N
- InChI
- 1S/C9H9BrO/c1-7-2-4-8(5-3-7)9(11)6-10/h2-5H,6H2,1H3
-
8-甲氧基补骨脂素分析标准品 ? 分析标准品 —— 纯度认证的材料,供定量校准使用。用于配制校准标准并验证分析方法。 Moligand™ ? Moligand™ —— 阿拉丁的配体和生物活性小分子系列。适用于需要明确小分子工具的受体、通路和结合研究。 ≥98%有现货 货号: M115185查看产品价格与包装
技术标识符
- IUPAC名称
- 9-methoxyfuro[3,2-g]chromen-7-one
- SMILES
- COC1=C2C(=CC3=C1OC=C3)C=CC(=O)O2
- InChIKey
- QXKHYNVANLEOEG-UHFFFAOYSA-N
- InChI
- 1S/C12H8O4/c1-14-12-10-8(4-5-15-10)6-7-2-3-9(13)16-11(7)12/h2-6H,1H3
-
2,4-二羟基苯甲酸甲酯有现货 货号: M117626查看产品价格与包装
技术标识符
- IUPAC名称
- methyl 2,4-dihydroxybenzoate
- SMILES
- COC(=O)C1=C(C=C(C=C1)O)O
- InChIKey
- IIFCLXHRIYTHPV-UHFFFAOYSA-N
- InChI
- 1S/C8H8O4/c1-12-8(11)6-3-2-5(9)4-7(6)10/h2-4,9-10H,1H3
-
4-(4-甲基哌嗪)苯胺有现货 货号: M121860查看产品价格与包装
技术标识符
- IUPAC名称
- 4-(4-methylpiperazin-1-yl)aniline
- SMILES
- CN1CCN(CC1)C2=CC=C(C=C2)N
- InChIKey
- MOZNZNKHRXRLLF-UHFFFAOYSA-N
- InChI
- 1S/C11H17N3/c1-13-6-8-14(9-7-13)11-4-2-10(12)3-5-11/h2-5H,6-9,12H2,1H3
-
MLN120B,IkappaB 激酶β (IKKβ) 抑制剂有现货 货号: M127370查看产品价格与包装
技术标识符
- IUPAC名称
- N-(6-chloro-7-methoxy-9H-pyrido[3,4-b]indol-8-yl)-2-methylpyridine-3-carboxamide
- SMILES
- CC1=C(C=CC=N1)C(=O)NC2=C3C(=CC(=C2OC)Cl)C4=C(N3)C=NC=C4
- InChIKey
- ZNOLRTPMNMPLHY-UHFFFAOYSA-N
- InChI
- 1S/C19H15ClN4O2/c1-10-11(4-3-6-22-10)19(25)24-17-16-13(8-14(20)18(17)26-2)12-5-7-21-9-15(12)23-16/h3-9,23H,1-2H3,(H,24,25)
-
莫特塞尼有现货 货号: M126795查看产品价格与包装
技术标识符
- IUPAC名称
- N-(3,3-dimethyl-1,2-dihydroindol-6-yl)-2-(pyridin-4-ylmethylamino)pyridine-3-carboxamide
- SMILES
- CC1(CNC2=C1C=CC(=C2)NC(=O)C3=C(N=CC=C3)NCC4=CC=NC=C4)C
- InChIKey
- RAHBGWKEPAQNFF-UHFFFAOYSA-N
- InChI
- 1S/C22H23N5O/c1-22(2)14-26-19-12-16(5-6-18(19)22)27-21(28)17-4-3-9-24-20(17)25-13-15-7-10-23-11-8-15/h3-12,26H,13-14H2,1-2H3,(H,24,25)(H,27,28)
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马赛替尼 (AB1010)CAS: 790299-79-5 分子式: C28H30N6OS 分子量: 498.65有现货 货号: M126981查看产品价格与包装
技术标识符
- IUPAC名称
- 4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[(4-pyridin-3-yl-1,3-thiazol-2-yl)amino]phenyl]benzamide
- SMILES
- CC1=C(C=C(C=C1)NC(=O)C2=CC=C(C=C2)CN3CCN(CC3)C)NC4=NC(=CS4)C5=CN=CC=C5
- InChIKey
- WJEOLQLKVOPQFV-UHFFFAOYSA-N
- InChI
- 1S/C28H30N6OS/c1-20-5-10-24(16-25(20)31-28-32-26(19-36-28)23-4-3-11-29-17-23)30-27(35)22-8-6-21(7-9-22)18-34-14-12-33(2)13-15-34/h3-11,16-17,19H,12-15,18H2,1-2H3,(H,30,35)(H,31,32)
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Amuvatinib (MP-470),抑制剂CAS: 850879-09-3 分子式: C23H21N5O3S 分子量: 447.52有现货 货号: M127412查看产品价格与包装
技术标识符
- IUPAC名称
- N-(1,3-benzodioxol-5-ylmethyl)-4-([1]benzofuro[3,2-d]pyrimidin-4-yl)piperazine-1-carbothioamide
- SMILES
- C1CN(CCN1C2=NC=NC3=C2OC4=CC=CC=C43)C(=S)NCC5=CC6=C(C=C5)OCO6
- InChIKey
- FOFDIMHVKGYHRU-UHFFFAOYSA-N
- InChI
- 1S/C23H21N5O3S/c32-23(24-12-15-5-6-18-19(11-15)30-14-29-18)28-9-7-27(8-10-28)22-21-20(25-13-26-22)16-3-1-2-4-17(16)31-21/h1-6,11,13H,7-10,12,14H2,(H,24,32)
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最后更新:2026年11月5日
如何使用蛋白激酶(Protein kinases)分类?
可用蛋白激酶(Protein kinases)快速圈定靶点范围,再逐一在各产品页面确认化合物信息。通路注释是导航辅助,不能替代对活性检测方法的核实。
蛋白激酶(Protein kinases)下收录了哪些靶点?
蛋白激酶(Protein kinases)包括丝裂原活化蛋白激酶1(MAPK1)、丙酮酸激酶 pkm (PKM)、丝氨酸蛋白激酶 atm (ATM)、表皮生长因子受体(EGFR)、糖原合成酶激酶-3β (GSK3B)等,另有508个子类别。选择某一靶点即可查看针对该靶点注释的抑制剂、激动剂和工具化合物。
从蛋白激酶(Protein kinases)订购化合物前应核查什么?
对于蛋白激酶(Protein kinases)中的任何化合物,请核查所报道活性的检测方法、对同家族相关靶点的选择性、纯度,以及推荐的母液溶剂和储存条件。批次数据见分析证书。所有产品仅供专业研发用途,不得用于人体、动物、诊断或治疗。
可以按作用机制筛选蛋白激酶(Protein kinases)化合物吗?
可以——您可在蛋白激酶(Protein kinases)中按靶点、作用机制和化合物类别筛选,并按靶点名称或基因符号、CAS号或SMILES搜索。大包装或未收录产品请联系 compliance@aladdinsci.com。












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