DNMT3A-IN-1 is a potent and selective DNMT3A inhibitor. DNMT3A-IN-1 shows inhibitor activities against DNMT3A with k I values range from 9.16-18.85 μM (AdoMet) and 11.37-23.34 μM (poly dI-dC)
Form:Solid
IC50& Target:DNMT3A
规格
规格或纯度
≥98%
英文名称
DNMT3A-IN-1
生化机理
DNMT3A-IN-1 是一种强效的 DNMT3A 选择性抑制剂。DNMT3A-IN-1 对 DNMT3A 具有抑制活性,其 k I 值范围为 9.16-18.85 μM(AdoMet)和 11.37-23.34 μM(poly dI-dC)。