ELA-21 (human) is an apelin receptor agonist with a pK i of 8.52. ELA-21 (human) completely inhibits Forskolin-induced cAMP production and stimulates β-arrestin recruitment with subnanomolar potencies. ELA-21 (human) is an agonist in G-protein-dependent and -independent pathways.
Form:Solid
规格
别名
ELA-21(人类)
规格或纯度
≥98%
英文名称
ELA-21 (human)
生化机理
ELA-21 (人)是一种 pK i 为 8.52 的芹菜素受体激动剂。ELA-21 (人)能完全抑制福斯可林诱导的 cAMP 生成,并以亚纳摩尔的效力刺激 β-restin 募集。ELA-21(人)是一种 G 蛋白依赖性 a