KNT-127 is a potent and selective δ-opioid receptor agonist effective by systemic administration. KNT-127 shows selectivity for the δ-receptor ( K i 0f 21.3, 0.16, 153 nM for opioid μ-, δ-, and κ-receptors, respectively). KNT-127 increases the release of dopamine and L-glutamate in the striatum, nucleus accumbens and median pre-frontal cortex. Antidepressant-like effects.
Form:Solid
规格
规格或纯度
≥99%
英文名称
KNT-127
生化机理
KNT-127 是一种强效的选择性δ-阿片受体激动剂,全身给药有效。KNT-127 对δ受体具有选择性(对阿片μ受体、δ受体和κ受体的 K i 0f 分别为 21.3、0.16 和 153 nM)。KNT-127 可增加阿片受体