Lei-Dab7 TFA is a high affinity, selective K Ca 2.2 (SK2) channel blocker (K d =3.8 nM). Lei-Dab7 TFA exhibits >200-fold selectivity for K Ca 2.2 over K Ca 2.1, K Ca 2.3, K Ca 3.1, K v and Kir2.1. Lei-Dab7 TFA increases theta-burst responses and increases
Appearance:Solid
Biological Activity:Lei-Dab7 TFA is a high affinity, selective K Ca 2.2 (SK2) channel blocker (K d =3.8 nM). Lei-Dab7 TFA exhibits >200-fold selectivity for K Ca 2.2 over K Ca 2.1, K Ca 2.3, K Ca 3.1, K v and Kir2.1. Lei-Dab7 TFA increases theta-burst responses and increases