MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan is a agent-linker conjugates for ADC , consisting Exatecan . Exatecan is a DNA Topoisomerase I inhibitor (IC 50 =2.2 μM)
Form:Solid
IC50& Target:Topoisomerase I
规格
别名
MC-Gly-Gly-Phe-Gly-(S)-环丙烷-依沙替康
规格或纯度
≥95%
英文名称
MC-Gly-Gly-Phe-Gly-(S)-Cyclopropane-Exatecan
生化机理
MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan是一种用于ADC的药剂连接体,由Exatecan(HY-13631)组成。Exatecan 是一种 DNA 拓扑异构酶 I 抑制剂(IC 50 =2.2 μM)。