Nociceptin (1-13), amide TFA is a potent ORL1 receptor (opioid receptor-like 1 receptor, OP4) agonist with a pEC 50 of 7.9 for mouse vas deferens and a K i of 0.75 nM for binding to rat forebrain membranes.
Appearance:Solid
IC50& Target:NOP Receptor/ORL1
Biological Activity:Nociceptin (1-13), amide TFA is a potent ORL1 receptor (opioid receptor-like 1 receptor, OP4) agonist with a pEC 50 of 7.9 for mouse vas deferens and a K i of 0.75 nM for binding to rat forebrain membranes .