PG106 TFA is a potent and selective human melanocortin 3 (hMC3) receptor antagonist ( IC 50 = 210 nM) and has noactivity at hMC4 receptors ( EC 50 =9900 nM) and hMC5 receptor.
Appearance:Solid
IC50& Target:MC3R
Biological Activity:PG106 TFA is a potent and selective human melanocortin 3 (hMC3) receptor antagonist ( IC 50 = 210 nM) and has noactivity atxa0hMC4xa0receptors ( EC 50 =9900 nM) andxa0hMC5xa0receptor.