(R)-Tegoprazan (example 3), a benzimidazole derivative, is a potent kidney H + /K + -ATPase inhibitor with an IC 50 of 98 nM of canine kidney Na + /K + -ATPase. (R)-Tegoprazan has the potential for gastrointestinal diseases research.
Form:Solid
规格
别名
(R)-替戈拉赞
规格或纯度
≥98%
英文名称
(R)-Tegoprazan
生化机理
(R)-Tegoprazan((R)-CJ-12420;例 3)是一种苯并咪唑衍生物,是一种强效的肾 H + /K + -ATPase 抑制剂,对犬肾 Na + /K + -ATPase 的 IC 50 为 98 nM。(R)-Tegoprazan 具有胃肠道疾病研究的潜力。