计算溶液所需的质量、体积或浓度。
提供 ≥99% 纯度,适用于对基线干扰要求严格的色谱和分析工作流程。
2-8°C储存。低温运输 。请查阅批次 COA 获取详细规格。
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在色谱分析、有机合成和交叉偶联反应领域已被 0 篇同行评审文献引用。
UNI418 is a dual inhibitor of PIKfyve and PIP5K1C with antiviral activity against SARS-CoV-2 ( EC 50 =1.4 μM). UNI418 blocks ACE2-mediated SARS-CoV-2 viral endocytosis by inhibiting PIP5K1C ( IC 50 =60.1 nM; K d =61 nM). In addition, UNI418 inhibits the proteolytic activation of proteases regulated by PIKfyve ( K d =0.78 nM) to prevent SARS-CoV-2 from entering host cells.